A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to a new dual alpha/gamma partial agonist endowed with mitochondrial pyruvate carrier inhibition and antidiabetic properties Article Swipe
Antonio Laghezza
,
Carmen Cerchia
,
Massimo Genovese
,
Roberta Montanari
,
Davide Capelli
,
Judith Wackerlig
,
Stefan Simić
,
Emanuele Falbo
,
Lucia Pecora
,
Rosalba Leuci
,
Leonardo Brunetti
,
Luca Piemontese
,
Paolo Tortorella
,
Abanish Biswas
,
Ravi Pratap Singh
,
Suhas Tambe
,
C A Sudeep
,
Ashok Pattnaik
,
Venkatesan Jayaprakash
,
Paolo Paoli
,
Antonio Lavecchia
,
Fulvio Loiodice
·
YOU?
·
· 2024
· Open Access
·
· DOI: https://doi.org/10.1016/j.ejmech.2024.116567
YOU?
·
· 2024
· Open Access
·
· DOI: https://doi.org/10.1016/j.ejmech.2024.116567
Related Topics
Concepts
Agonist
Partial agonist
Chemistry
In vivo
Pharmacology
Peroxisome proliferator-activated receptor
Receptor
PPAR agonist
In vitro
Endocrinology
Biochemistry
Internal medicine
Biology
Medicine
Biotechnology
Metadata
- Type
- article
- Language
- en
- Landing Page
- https://doi.org/10.1016/j.ejmech.2024.116567
- OA Status
- green
- Cited By
- 3
- References
- 56
- Related Works
- 10
- OpenAlex ID
- https://openalex.org/W4399471952
All OpenAlex metadata
Raw OpenAlex JSON
- OpenAlex ID
-
https://openalex.org/W4399471952Canonical identifier for this work in OpenAlex
- DOI
-
https://doi.org/10.1016/j.ejmech.2024.116567Digital Object Identifier
- Title
-
A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to a new dual alpha/gamma partial agonist endowed with mitochondrial pyruvate carrier inhibition and antidiabetic propertiesWork title
- Type
-
articleOpenAlex work type
- Language
-
enPrimary language
- Publication year
-
2024Year of publication
- Publication date
-
2024-06-09Full publication date if available
- Authors
-
Antonio Laghezza, Carmen Cerchia, Massimo Genovese, Roberta Montanari, Davide Capelli, Judith Wackerlig, Stefan Simić, Emanuele Falbo, Lucia Pecora, Rosalba Leuci, Leonardo Brunetti, Luca Piemontese, Paolo Tortorella, Abanish Biswas, Ravi Pratap Singh, Suhas Tambe, C A Sudeep, Ashok Pattnaik, Venkatesan Jayaprakash, Paolo Paoli, Antonio Lavecchia, Fulvio LoiodiceList of authors in order
- Landing page
-
https://doi.org/10.1016/j.ejmech.2024.116567Publisher landing page
- Open access
-
YesWhether a free full text is available
- OA status
-
greenOpen access status per OpenAlex
- OA URL
-
https://hdl.handle.net/11586/485320Direct OA link when available
- Concepts
-
Agonist, Partial agonist, Chemistry, In vivo, Pharmacology, Peroxisome proliferator-activated receptor, Receptor, PPAR agonist, In vitro, Endocrinology, Biochemistry, Internal medicine, Biology, Medicine, BiotechnologyTop concepts (fields/topics) attached by OpenAlex
- Cited by
-
3Total citation count in OpenAlex
- Citations by year (recent)
-
2025: 2, 2024: 1Per-year citation counts (last 5 years)
- References (count)
-
56Number of works referenced by this work
- Related works (count)
-
10Other works algorithmically related by OpenAlex
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