Novel specific activity-based probes validate KLK proteases as druggable targets Article Swipe

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Georgia Sotiropoulou , Eleni Zingkou , Georgios Pampalakis ·

YOU? · · 2022 · Open Access · · DOI: https://doi.org/10.1080/15384047.2022.2074775

KEYWORDS: activity-based probesABPskallikrein-related peptidasesKLKsKLK-ABPsKLK proteolytic cascadesactivographytheranostic ABPs

Related Topics

Computational Biology

Biology

Biochemistry

Concepts

Druggability Proteases Computational biology Biology Cancer research Biochemistry Enzyme Gene

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Type: letter
Language: en
Landing Page: https://doi.org/10.1080/15384047.2022.2074775
PDF: https://www.tandfonline.com/doi/pdf/10.1080/15384047.2022.2074775?needAccess=true
OA Status: gold
References: 25
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DOI: https://doi.org/10.1080/15384047.2022.2074775

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Title: Novel specific activity-based probes validate KLK proteases as druggable targets

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Type: letter

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Language: en

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Publication year: 2022

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Publication date: 2022-06-02

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Authors: Georgia Sotiropoulou, Eleni Zingkou, Georgios Pampalakis

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Landing page: https://doi.org/10.1080/15384047.2022.2074775

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PDF URL: https://www.tandfonline.com/doi/pdf/10.1080/15384047.2022.2074775?needAccess=true

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OA URL: https://www.tandfonline.com/doi/pdf/10.1080/15384047.2022.2074775?needAccess=true

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Concepts: Druggability, Proteases, Computational biology, Biology, Cancer research, Biochemistry, Enzyme, Gene

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Cited by: 0

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References (count): 25

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