Anjie S. Bispat
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View article: Inhibition of N-type calcium channels by phenoxyaniline and sulfonamide analogues
Inhibition of N-type calcium channels by phenoxyaniline and sulfonamide analogues Open
A detailed SAR study led to two potent Ca V 2.2 inhibitors, the sulfonamide derivatives 42 and 45, which showed high plasma stability, low toxicity, favourable CNS MPO scores (4.0–4.4), and strong potency.
View article: The neuronal calcium ion channel activity of constrained analogues of MONIRO-1
The neuronal calcium ion channel activity of constrained analogues of MONIRO-1 Open
View article: Synthesis and evaluation of aminobenzothiazoles as blockers of N- and T-type calcium channels
Synthesis and evaluation of aminobenzothiazoles as blockers of N- and T-type calcium channels Open